TargetMol

ZEN-3411

Product Code:
 
TAR-T13393
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T13393-5mg5mg£850.00
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Quantity:
TAR-T13393-50mg50mg£1,661.00
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Quantity:
TAR-T13393-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
ZEN-3411 is an inhibitor of BET(IC50s of 0.05, 0.05 and 0.06 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively). ZEN-3411 can be used to form PROTACs to induce degradation of BRD4.
CAS:
1952264-36-6
Formula:
C21H20N4O2
Molecular Weight:
360.417
Pathway:
Proteases/Proteasome
Purity:
0.98
SMILES:
Cc1noc(C)c1-c1cc(N)c2ncn(Cc3ccc(cc3)C3CO3)c2c1
Target:
Serine Protease

References

1. Kharenko OA, et al. Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain (BET) Inhibitors Targeting a Methionine. J Med Chem. 2018 Sep 27;61(18):8202-8211.