CGRP antagonist 1

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TargetMol
Product Code: TAR-T13453
Supplier: TargetMol
CodeSizePrice
TAR-T13453-1mg1mg£345.00
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TAR-T13453-5mg5mg£736.00
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TAR-T13453-10mg10mg£994.00
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Quantity:
TAR-T13453-25mg25mg£1,420.00
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Quantity:
TAR-T13453-50mg50mg£1,910.00
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Quantity:
TAR-T13453-100mg100mg£2,456.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
CGRP antagonist 1 is a highly potent antagonist of CGRP receptor(Ki and IC50 of 35 and 57 nM, respectively).
CAS:
1123757-49-2
Formula:
C29H26N4O4
Molecular Weight:
494.551
Pathway:
Metabolism
Purity:
0.98
SMILES:
O=C(CN1C(=O)C2(CCOCC2)c2ccccc12)Nc1ccc2C[C@@]3(Cc2c1)C(=O)Nc1ncccc31
Target:
Dehydrogenase

References

1. Stump CA, et al. The discovery of highly potent CGRP receptor antagonists. Bioorg Med Chem Lett. 2009 Jan 1;19(1):214-7.