BETd-246

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TargetMol
Product Code: TAR-T14549
Supplier: TargetMol
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TAR-T14549-100mg100mgEnquire
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TAR-T14549-5mg5mg£503.00
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TAR-T14549-10mg10mg£704.00
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TAR-T14549-50mg50mg£2,030.00
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Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
BETd-246 is an inhibitor of second-generation and PROTAC-based BET bromodomain (BRD), show antitumor activity.
CAS:
2140289-17-2
Formula:
C48H55N11O10
Molecular Weight:
946.035
Purity:
0.98
SMILES:
CCn1nc(cc1Nc1nc(nc2[nH]c3cc(-c4c(C)noc4C)c(OC)cc3c12)C(=O)NCCCOCCOCCOCCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12)C1CC1

References

1. Bai L, et al. Targeted Degradation of BET Proteins in Triple-Negative Breast Cancer. Cancer Res. 2017 May 1;77(9):2476-2487.