Varespladib

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TargetMol
Product Code: TAR-T2044
Supplier: TargetMol
CodeSizePrice
TAR-T2044-1mg1mg£101.00
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TAR-T2044-2mg2mg£114.00
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TAR-T2044-5mg5mg£142.00
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Quantity:
TAR-T2044-1mL1 mL * 10 mM (in DMSO)£173.00
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TAR-T2044-10mg10mg£195.00
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TAR-T2044-25mg25mg£322.00
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TAR-T2044-50mg50mg£466.00
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TAR-T2044-100mg100mg£651.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
Varespladib, a specific and effective human non-pancreatic secretory phospholipase A2 (hnsPLA) inhibitor(IC50=7 nM), has been investigated for the treatment and prevention of sickle cell disease, vaso-occlusive crisis, and acute coronary syndrome.
CAS:
172732-68-2
Formula:
C21H20N2O5
Molecular Weight:
380.4
Pathway:
Metabolism
Purity:
0.98
SMILES:
CCc1c(C(=O)C(N)=O)c2c(OCC(O)=O)cccc2n1Cc1ccccc1
Target:
Phospholipase

References

1. Draheim SE, et al. J Med Chem. 1996, 39(26), 5159-5175. 2. Snyder DW, et al. J Pharmacol Exp Ther. 1999, 288(3), 1117-1124. 3. Hori Y, et al. Invest Ophthalmol Vis Sci. 2005, 46(11), 4050-4061.