EHop-016

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TargetMol
Product Code: TAR-T2427
Supplier: TargetMol
CodeSizePrice
TAR-T2427-5mg5mg£103.00
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TAR-T2427-1mL1 mL * 10 mM (in DMSO)£106.00
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TAR-T2427-10mg10mg£124.00
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TAR-T2427-25mg25mg£174.00
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TAR-T2427-50mg50mg£251.00
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Quantity:
TAR-T2427-100mg100mg£389.00
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TAR-T2427-200mg200mg£538.00
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TAR-T2427-500mg500mg£804.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
EHop-016 is a specific Rac GTPase inhibitor with IC50 of 1.1 μM for Rac1 in MDA-MB-231 and MDA-MB-435 cells, equally effective inhibition for Rac3.
CAS:
1380432-32-5
Formula:
C25H30N6O
Molecular Weight:
430.556
Pathway:
GPCR/G Protein; Cell Cycle/Checkpoint; MAPK
Purity:
0.9769
SMILES:
CCn1c2ccccc2c2cc(Nc3ccnc(NCCCN4CCOCC4)n3)ccc12
Target:
Rho; Ras

References

1. Montalvo-Ortiz BL, et al. J Biol Chem. 2012, 287(16), 13228-13238. 2. Martin H, et al. J Clin Invest. 2013, 123(10), 4449-4463.