L 366948
Code | Size | Price |
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TAR-T24292-5mg | 5mg | £1,010.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T24292-50mg | 50mg | £1,982.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T24292-100mg | 100mg | £2,560.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
L 366948 is an antagonist of the oxytocin receptor.
CAS:
127819-97-0
Formula:
C42H54N8O6
Molecular Weight:
766.944
Purity:
0.98
SMILES:
CCC(C)C1NC(=O)C(Cc2ccc3ccccc3c2)NC(=O)C2CCCN2C(=O)C(Cc2cnc[nH]2)NC(=O)C2CCCCN2C(=O)C2CCCCN2C1=O
References
1. Politowska E, Drabik P, Kazmierkiewicz R, Ciarkowsk J. Docking ligands to vasopressin and oxytocin receptors via genetic algorithm. J Recept Signal Transduct Res. 2002 Feb-Nov;22(1-4):393-409. PubMed PMID: 12503629.
2. Hu J, Ludwig TE, Salli U, Stormshak F, Mirando MA. Autocrine/paracrine action of oxytocin in pig endometrium. Biol Reprod. 2001 Jun;64(6):1682-8. PubMed PMID: 11369595.
3. Politowska E, Czaplewski C, Ciarkowski J. Molecular modeling of the oxytocin receptor/bioligand interactions. Acta Biochim Pol. 1999;46(3):581-90. PubMed PMID: 10698266.
4. Yibchok-Anun S, Cheng H, Heine PA, Hsu WH. Characterization of receptors mediating AVP- and OT-induced glucagon release from the rat pancreas. Am J Physiol. 1999 Jul;277(1 Pt 1):E56-62. PubMed PMID: 10409128.