CPI203

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TargetMol
Product Code: TAR-T2442
Supplier: TargetMol
CodeSizePrice
TAR-T2442-1mL1 mL * 10 mM (in DMSO)£111.00
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TAR-T2442-5mg5mg£111.00
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Quantity:
TAR-T2442-10mg10mg£131.00
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Quantity:
TAR-T2442-25mg25mg£167.00
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Quantity:
TAR-T2442-50mg50mg£248.00
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Quantity:
TAR-T2442-100mg100mg£390.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
CPI-203 is an effective BET bromodomain inhibitor (IC50: 37 nM for BRD4).
CAS:
202591-23-9
Formula:
C19H18ClN5OS
Molecular Weight:
399.9
Pathway:
Chromatin/Epigenetic
Purity:
0.9913
SMILES:
Cc1nnc2C(CC(N)=O)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1
Target:
Epigenetic Reader Domain

References

1. Devaiah BN, et al. Proc Natl Acad Sci U S A. 2012, 109(18), 6927-6932. 2. Moros A, et al. Leukemia. 2014. doi: 10.1038/leu.2014.106.