APTAA-LHRH
| Code | Size | Price |
|---|
| TAR-T25105-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Documents
Further Information
Bioactivity:
APTAA-LHRH is a gonadorelin antagonist.
CAS:
83539-08-6
Formula:
C69H91Cl2N17O14
Molecular Weight:
1453.49
Purity:
0.98
SMILES:
CC(C)C[C@H](NC(=O)[C@@H](CCCNC(N)=N)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CO)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](Cc1ccc(Cl)cc1)NC(=O)[C@@H](Cc1ccc(Cl)cc1)NC(C)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N1CCC[C@H]1C(=O)N[C@H](C)C(O)=O
References
1. van den Dungen HM, Dijkstra H, Hiehle MA, van Rees GP, Schoemaker J. Effects of LHRH antagonist administration to immature male rats on sexual development. Physiol Behav. 1989 Nov;46(5):779-85. PubMed PMID: 2516908.
2. Deckers GH, de Graaf JH, Kloosterboer HJ, Loozen HJ. Properties of a potent LHRH antagonist (Org 30850) in female and male rats. J Steroid Biochem Mol Biol. 1992 Aug;42(7):705-12. PubMed PMID: 1504009.
3. Geisthoevel F, Arana JB, Balmaceda JP, Rojas FJ, Asch RH. Prolactin and gonadotrophin dynamics in response to antagonists of LHRH and dopamine in ovariectomized rhesus monkeys: a dissection of their common secretion. Hum Reprod. 1988 Jul;3(5):591-5. PubMed PMID: 3139699.
4. S?nchez-Criado JE, Hernandez G, Bellido C, Gonzalez D, T?bar M, Diaz-Cruz MA, Alonso R. Periovulatory LHRH, LH and FSH secretion in cyclic rats treated with RU486: effects of exogenous LHRH and LHRH antagonist on LH and FSH secretion at early oestrus. J Endocrinol. 1994 Apr;141(1):7-14. PubMed PMID: 8014605.