Boc-ypgflt(O-tbu)
| Code | Size | Price |
|---|
| TAR-T25168-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Documents
Further Information
Bioactivity:
Boc-ypgflt(O-tbu) is a delta-receptor-selective opioid antagonist.
CAS:
179124-36-8
Formula:
C44H64N6O11
Molecular Weight:
853.027
Purity:
0.98
SMILES:
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H]([C@@H](C)OC(C)(C)C)C(O)=O
References
1. R?nai AZ, Magyar A, Orosz G, Borsodi A, Benyhe S, T?th G, Mak? E, K?tay E, Babka E, Medzihradszky K. Opioid antagonist properties of the highly delta-receptor-selective BOC-Tyr-Pro-Gly-Phe-Leu-Thr (OtBu) peptide and of its Phe1 and Mel1 analogues. Arch Int Pharmacodyn Ther. 1995 Nov-Dec;330(3):361-9. PubMed PMID: 8836454.
2. Mak? E, R?nai AZ, Ad?m G, Juh?sz G, Ritter L, Lest?r B, Crunelli V. Modulation by GABA(B) and delta opioid receptors of neurally induced responses in isolated guinea-pig taenia coli and human colonic circular muscle. J Physiol Paris. 2000 Mar-Apr;94(2):135-8. PubMed PMID: 10791695.