Levallorphan tartrate

TargetMol
Product Code: TAR-T25690
Supplier: TargetMol
CodeSizePrice
TAR-T25690-5mg5mg£850.00
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Quantity:
TAR-T25690-50mg50mg£1,661.00
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Quantity:
TAR-T25690-100mg100mg£2,079.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Further Information

Bioactivity:
Levallorphan tartrate is an opioid antagonist with properties similar to those of NALOXONE. Levallorphan reverses severe opioid-induced respiratory depression but may exacerbate respiratory depression such as that induced by alcohol or other non-opioid central depressants.
CAS:
71-82-9
Formula:
C23H31NO7
Molecular Weight:
433.501
Purity:
0.98
SMILES:
O[C@H]([C@@H](O)C(O)=O)C(O)=O.[H][C@@]12CCCC[C@@]11CCN(CC=C)[C@@H]2Cc2ccc(O)cc12

References

1. MILLER JW, GILFOIL TM, SHIDEMAN FE. The effects of levallorphan tartrate (levo-3-hydroxy-N-allylmorphinan tartrate) on the respiration of rabbits given morphine. J Pharmacol Exp Ther. 1955 Nov;115(3):350-9. PubMed PMID: 13272187. 2. GRUBER CM Jr. Effect of levallorphan tartrate upon toxicity of morphine. Proc Soc Exp Biol Med. 1955 Feb;88(2):189-91. PubMed PMID: 14357383. 3. RANKIN J, MEHNERT J, CURRERI AR. Effect of levallorphan tartrate on levorphanol tartrate analgesia in postoperative patients. AMA Arch Surg. 1957 Apr;74(4):602-5. PubMed PMID: 13410340. 4. SCHNIEDEN H. The effect of levallorphan tartrate and of adiphenine hydrochloride on the antidiuretic action of morphine and nicotine. Br J Pharmacol Chemother. 1960 Dec;15:510-2. PubMed PMID: 13748312; PubMed Central PMCID: PMC1482260.