Phelorphan
Code | Size | Price |
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TAR-T25941-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T25941-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T25941-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Phelorphan is an inhibitor of enkephalinase.
CAS:
110871-16-4
Formula:
C20H22N2O4S
Molecular Weight:
386.47
Purity:
0.98
SMILES:
OC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)CS
References
1. Van Amsterdam JG, Llorens-Cortes C. Inhibition of enkephalin degradation by phelorphan: effects on striatal [Met5]enkephalin levels and jump latency in mouse hot plate test. Eur J Pharmacol. 1988 Sep 23;154(3):319-24. PubMed PMID: 3234484.
2. Haffmans J, Walsum MV, van Amsterdam JC, Dzoljic MR. Phelorphan, an inhibitor of enzymes involved in the biodegradation of enkephalins, affected the withdrawal symptoms in chronic morphine-dependent rats. Neuroscience. 1987 Jul;22(1):233-6. PubMed PMID: 2888045.
3. van Amsterdam JG, van Buuren KJ, Krielaart MJ, Zuiderveld OP, Tijms RP. Effect of inhibitors of enkephalin degradation in the isolated guinea-pig ileum. Life Sci. 1988;43(19):1529-36. PubMed PMID: 3193845.
4. Dzoljic MR. Enkephalinase inhibitors attenuate naloxone-precipitated withdrawal syndrome. NIDA Res Monogr. 1986;75:575-8. PubMed PMID: 3123978.