TargetMol

RGH 1756

Product Code:
 
TAR-T26069
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T26069-5mg5mg£850.00
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TAR-T26069-50mg50mg£1,661.00
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Quantity:
TAR-T26069-100mg100mg£2,079.00
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This product comes from: United States.
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  • Further Information
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Further Information

Bioactivity:
RGH 1756 is an atypical antipsychotic with high affinity to dopamine D(3) receptors that leads to c-Fos induction in a unique pattern.
CAS:
207277-37-0
Formula:
C26H30N4O2S
Molecular Weight:
462.61
Purity:
0.98
SMILES:
COc1ccccc1N1CCN(CCCCOc2ccc(cc2)-c2cn3ccsc3n2)CC1

References

1. G?mesi LI, Kap?s M, Szeber?nyi S. Application of LC-MS analysis to the characterisation of the in vitro and in vivo metabolite profiles of RGH-1756 in the rat. J Pharm Biomed Anal. 2001 Mar;24(5-6):877-85. PubMed PMID: 11248481. 2. Kov?cs KJ, Csejtei M, Laszlovszky I. Double activity imaging reveals distinct cellular targets of haloperidol, clozapine and dopamine D(3) receptor selective RGH-1756. Neuropharmacology. 2001 Mar;40(3):383-93. PubMed PMID: 11166331. 3. S?v?g? J, Farde L, Halldin C, Schukin E, Schou M, Laszlovszky I, Kiss B, Guly?s B. Lack of effect of reserpine-induced dopamine depletion on the binding of the dopamine-D3 selective radioligand, [11C]RGH-1756. Brain Res Bull. 2005 Oct 15;67(3):219-24. PubMed PMID: 16144658. 4. Terj?ki E, Kap?s M. An HPLC/UV method for the determination of RGH-1756 in dog and rat plasma. J Pharm Biomed Anal. 2001 Mar;24(5-6):913-20. PubMed PMID: 11248484.