GSK429286A

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TargetMol
Product Code: TAR-T2633
Supplier: TargetMol
CodeSizePrice
TAR-T2633-2mg2mg£99.00
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TAR-T2633-5mg5mg£115.00
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TAR-T2633-1mL1 mL * 10 mM (in DMSO)£121.00
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TAR-T2633-10mg10mg£139.00
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TAR-T2633-25mg25mg£182.00
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TAR-T2633-50mg50mg£243.00
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TAR-T2633-100mg100mg£367.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
GSK429286A is a specific inhibitor of ROCK1/2 (IC50: 14/63 nM).
CAS:
864082-47-3
Formula:
C21H16F4N4O2
Molecular Weight:
432.379
Pathway:
Cell Cycle/Checkpoint; Stem Cells; Cytoskeletal Signaling
Purity:
0.9842
SMILES:
CC1=C(C(CC(=O)N1)c1ccc(cc1)C(F)(F)F)C(=O)Nc1cc2cn[nH]c2cc1F
Target:
ROCK

References

1. Goodman KB, et al. J Med Chem, 2007, 50(1), 6-9. 2. Nichols RJ, et al. Biochem J, 2009, 424(1), 47-60.