2-AEMP TFA

TargetMol
Product Code: TAR-T26380
Supplier: TargetMol
CodeSizePrice
TAR-T26380-5mg5mg£246.00
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Quantity:
TAR-T26380-25mg25mg£525.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Further Information

Bioactivity:
2-AEMP TFA is a potent and rapidly acting antagonist of GABA(A)-?1 receptors. 2-AEMP is an analog of GABA.
CAS:
321882-95-5
Formula:
C5H10F3NO5P
Molecular Weight:
252.107
Purity:
0.98
SMILES:
OC(=O)C(F)(F)F.CP([O-])(=O)OCCN

References

1. Xie A, Yan J, Yue L, Feng F, Mir F, Abdel-Halim H, Chebib M, Le Breton GC, Standaert RF, Qian H, Pepperberg DR. 2-Aminoethyl methylphosphonate, a potent and rapidly acting antagonist of GABA(A)-?1 receptors. Mol Pharmacol. 2011 Dec;80(6):965-78. doi: 10.1124/mol.111.071225. Epub 2011 Aug 2. PubMed PMID: 21810922; PubMed Central PMCID: PMC3228531. 2. Wang J, Mojumder DK, Yan J, Xie A, Standaert RF, Qian H, Pepperberg DR, Frishman LJ. In vivo electroretinographic studies of the role of GABAC receptors in retinal signal processing. Exp Eye Res. 2015 Oct;139:48-63. doi: 10.1016/j.exer.2015.07.002. Epub 2015 Jul 8. PubMed PMID: 26164072; PubMed Central PMCID: PMC4573340.