A 75998
| Code | Size | Price |
|---|
| TAR-T26443-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
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Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Documents
Further Information
Bioactivity:
A 75998 is a synthetic antagonist of leuteinizing hormone releasing hormone.
CAS:
135215-95-1
Formula:
C82H110ClN15O15
Molecular Weight:
1581.32
Purity:
0.98
SMILES:
CC(O)=O.CC(C)C[C@H](NC(=O)[C@H](CCCCNCc1cccnc1)NC(=O)[C@H](Cc1ccc(O)cc1)N(C)C(=O)[C@H](CO)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(Cl)cc1)C(=O)N([C@@H](C)C(=O)C(CC[C@H](NC(C)=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](C)C(=O)Nc1cccnc1)CNC(C)C)c1ccc2ccccc2c1
References
1. Haviv F, Bush EN, Knittle J, Greer J. LHRH antagonists. Pharm Biotechnol. 1998;11:131-49. Review. PubMed PMID: 9760679.
2. Cannon JB, Krill SL, Porter WR. Physicochemical properties of A-75998, an antagonist of luteinizing hormone releasing hormone. J Pharm Sci. 1995 Aug;84(8):953-8. PubMed PMID: 7500280.
3. Haviv F, Fitzpatrick TD, Nichols CJ, Bush EN, Diaz G, Bammert G, Nguyen AT, Johnson ES, Knittle J, Greer J. In vitro and in vivo activities of reduced-size antagonists of luteinizing hormone-releasing hormone. J Med Chem. 1994 Mar 4;37(5):701-5. PubMed PMID: 7510341.