TargetMol

A 81282

Product Code:
 
TAR-T26453
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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TAR-T26453-5mg5mg£850.00
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Further Information

Bioactivity:
A 81282 is a selective antagonist of angiotensin receptors. It has the activity of lowering blood pressure.
CAS:
141872-46-0
Formula:
C23H23N7O2
Molecular Weight:
429.484
Purity:
0.98
SMILES:
CCCCN(Cc1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1ncncc1C(O)=O

References

1. Hancock AA, Buckner SA, Lee JY, Brune M, Morse PA, Oheim K, Warner RB, Winn M, Zydowsky TM, De B, et al. Pharmacological characterization of Abbott-81282, a novel, non-peptide angiotensin-II antagonist selective for type-1 receptors. Life Sci. 1993;53(11):929-37. PubMed PMID: 8366760. 2. Lee JY, Brune ME, Warner RB, Buckner SB, Winn M, De B, Zydowsky TM, Opgenorth TJ, Kerkman DJ, DeBernardis JF. Antihypertensive activity of ABBOTT 81282, a nonpeptide angiotensin II antagonist, in the renal hypertensive rat. Pharmacology. 1993 Sep;47(3):176-87. PubMed PMID: 8415868.