Aza-THIP
Code | Size | Price |
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TAR-T26711-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T26711-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T26711-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Aza-THIP is a GABA-C-selective antagonist.
CAS:
654666-65-6
Formula:
C6H9N3O
Molecular Weight:
139.158
Purity:
0.98
SMILES:
Oc1n[nH]c2CNCCc12
References
1. Valembois S, Krall J, Fr?lund B, Steffansen B. Imidazole-4-acetic acid, a new lead structure for interaction with the taurine transporter in outer blood-retinal barrier cells. Eur J Pharm Sci. 2017 May 30;103:77-84. doi: 10.1016/j.ejps.2017.02.041. Epub 2017 Mar 1. PubMed PMID: 28259832.
2. Johnston GA, Chebib M, Hanrahan JR, Mewett KN. Neurochemicals for the investigation of GABA(C) receptors. Neurochem Res. 2010 Dec;35(12):1970-7. doi: 10.1007/s11064-010-0271-7. Epub 2010 Oct 21. Review. PubMed PMID: 20963487.
3. Krehan D, Fr?lund B, Ebert B, Nielsen B, Krogsgaard-Larsen P, Johnston GA, Chebib M. Aza-THIP and related analogues of THIP as GABA C antagonists. Bioorg Med Chem. 2003 Nov 17;11(23):4891-6. PubMed PMID: 14604650.
4. Johnston GA, Chebib M, Hanrahan JR, Mewett KN. GABA(C) receptors as drug targets. Curr Drug Targets CNS Neurol Disord. 2003 Aug;2(4):260-8. Review. PubMed PMID: 12871036.