Bisaramil hydrochloride
Code | Size | Price |
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TAR-T26822-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T26822-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T26822-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
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Further Information
Bioactivity:
Bisaramil, a calcium channel antagonist and sodium channel antagonist, is used potentially for the treatment of arrhythmia.
CAS:
96480-44-3
Formula:
C17H24Cl2N2O2
Molecular Weight:
359.29
Purity:
0.98
SMILES:
Cl.CCN1C[C@@H]2CN(C)C[C@H](C1)[C@H]2OC(=O)c1ccc(Cl)cc1
References
1. Haruno A, Sugiyama A, Hashimoto K. Chronotropic, inotropic, dromotropic and coronary vasodilator effects of bisaramil, a new class I antiarrhythmic drug, assessed using canine isolated, blood-perfused heart preparations. Jpn J Pharmacol. 1999 Jul;80(3):267-70. PubMed PMID: 10461773.
2. Pugsley MK, Goldin AL. Effects of bisaramil, a novel class I antiarrhythmic agent, on heart, skeletal muscle and brain Na+ channels. Eur J Pharmacol. 1998 Jan 19;342(1):93-104. PubMed PMID: 9544797.
3. Par?czai M, R?th E, K?rp?ti E. Bisaramil and antiarrhythmics as inhibitors of free radical generation. Pharmacol Res. 1997 Apr;35(4):279-85. PubMed PMID: 9264043.
4. R?th E, Lantos J, Temes G, Varga G, Par?czai M, K?rp?ti E. Cardioprotection during heart ischemia-reperfusion. Acta Chir Hung. 1997;36(1-4):306-9. PubMed PMID: 9408384.