BMS-902483
Code | Size | Price |
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TAR-T26862-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T26862-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T26862-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
BMS-902483 is a potent α7 partial agonist. BMS-902483 improved cognition in preclinical rodent models. BMS-902483 showed FLIR α7 EC50=9.3nM; α7 Electrophysiology, rat; Area EC50 = 140 nM; Peak, Area (Ymax %) = 40, 54. 5-HT3A IC50 = 480 nm.
CAS:
1192810-88-0
Formula:
C18H20N4O
Molecular Weight:
308.385
Purity:
0.98
SMILES:
C1N=C(Nc2cc3ccccc3cn2)O[C@]11CN2CC[C@H]1CC2
References
1. Design and Synthesis of a New Series of 4-Heteroarylamino-1?-azaspiro[oxazole-5,3?-bicyclo[2.2.2]octanes as ?7 Nicotinic Receptor Agonists. 1. Development of Pharmacophore and Early Structure?Activity Relationship James CookF. MacorRichard E. Olson Publication Date (Web): November 18, 2016 (Article) doi: 10.1021/acs.jmedchem.6b01506