Bromerguride
Code | Size | Price |
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TAR-T26909-5mg | 5mg | £1,500.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T26909-50mg | 50mg | £6,480.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T26909-100mg | 100mg | £9,307.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Bromerguride is a dopamine antagonist with the activity of antipsychotic.
CAS:
83455-48-5
Formula:
C20H25BrN4O
Molecular Weight:
417.351
Purity:
0.98
SMILES:
[H][C@@]12Cc3c(Br)[nH]c4cccc(C1=C[C@@H](CN2C)NC(=O)N(CC)CC)c34
References
1. Hilderbrand M, H?mpel M, Krause W, T?uber U. Pharmacokinetics of bromerguride, a new dopamine-antagonistic ergot derivative in rat and dog. Eur J Drug Metab Pharmacokinet. 1987 Jan-Mar;12(1):31-40. PubMed PMID: 3609071.
2. Krause W, Sauerbrey N, Gr?f KJ. Pharmacokinetics and pharmacodynamics in man of the dopamine antagonist ergot derivative, bromerguride. Eur J Clin Pharmacol. 1986;31(2):165-8. PubMed PMID: 3803415.
3. Martinot JL, Paill?re-Martinot ML, Loc'h C, Hardy P, Poirier MF, Mazoyer B, Beaufils B, Mazi?re B, Allilaire JF, Syrota A. The estimated density of D2 striatal receptors in schizophrenia. A study with positron emission tomography and 76Br-bromolisuride. Br J Psychiatry. 1991 Mar;158:346-50. PubMed PMID: 1827999.
4. Assi? MB, Cosi C, Koek W. 5-HT1A receptor agonist properties of the antipsychotic, nemonapride: comparison with bromerguride and clozapine. Eur J Pharmacol. 1997 Sep 10;334(2-3):141-7. PubMed PMID: 9369342.