Cilansetron
Code | Size | Price |
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TAR-T27020-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T27020-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T27020-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Cilansetron is a 5-HT3 antagonist. Cilansetron antagonizes the sensitivity of mesenteric afferent fibres to 5-hydroxytryptamine in the rat jejunum.
CAS:
120635-74-7
Formula:
C20H21N3O
Molecular Weight:
319.408
Purity:
0.98
SMILES:
Cc1nccn1C[C@H]1CC=C2C(c3cccc4CCCN2c34)C1=O
References
1. Painsipp E, Shahbazian A, Holzer P. Alosetron, cilansetron and tegaserod modify mesenteric but not colonic blood flow in rats. Br J Pharmacol. 2009 Nov;158(5):1210-26. doi: 10.1111/j.1476-5381.2009.00392.x. Epub 2009 Sep 25. PubMed PMID: 19785647; PubMed Central PMCID: PMC2782331.
2. Stacher G. Cilansetron in the treatment of diarrhea-predominant irritable bowel syndrome? Expert Rev Gastroenterol Hepatol. 2007 Oct;1(1):15-27. doi: 10.1586/17474124.1.1.15. Review. PubMed PMID: 19072430.
3. Olden KW, Crowell MD. Cilansetron. Drugs Today (Barc). 2005 Oct;41(10):661-6. Review. PubMed PMID: 16389408.
4. Cilansetron: KC 9946. Drugs R D. 2005;6(3):169-73. Review. PubMed PMID: 15869320.