EO-122
Code | Size | Price |
---|
TAR-T27272-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T27272-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T27272-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
EO-122, a calcium channel antagonist and sodium channel antagonist, is used potentially for the treatment of arrhythmia.
CAS:
23581-62-6
Formula:
C16H23ClN2O
Molecular Weight:
294.82
Purity:
0.98
SMILES:
Cl.Cc1cccc(C)c1NC(=O)C1CN2CCC1CC2
References
1. Oppenheimer E, Harel G, Lipinsky D, Sarne Y. EO-199, a specific antagonist of antiarrhythmic drugs: assessment by binding experiments and in vivo studies. Life Sci. 1991;48(10):977-85. PubMed PMID: 2000027.
2. Oppenheimer E, Meiri H, Ori Y. The specific binding of [3H]EO-122, a radiolabeled class I antiarrhythmic drug to rat heart membranes. J Mol Cell Cardiol. 1989 Feb;21(2):223-30. Erratum in: J Mol Cell Cardiol 1989 Dec;21(12):1356. PubMed PMID: 2545887.
3. Marrer S. [Molecular modeling of anti-arrhythmia agents in class Ia and Ib--model conceptions of different binding receptors]. Pharm Acta Helv. 1989;64(12):338-44. German. PubMed PMID: 2616583.
4. Binah O, Gilat E, Rubinstein I, Oppenheimer E. Electrophysiological effects of a novel antiarrhythmic drug, EO-122, on guinea pig ventricular muscle and isolated myocytes. J Cardiovasc Pharmacol. 1987 Sep;10(3):301-8. PubMed PMID: 2444778.