GSK2008607

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TargetMol
Product Code: TAR-T27454
Supplier: TargetMol
CodeSizePrice
TAR-T27454-1mg1mg£352.00
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TAR-T27454-5mg5mg£736.00
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Quantity:
TAR-T27454-10mg10mg£978.00
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Quantity:
TAR-T27454-25mg25mg£1,348.00
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Quantity:
TAR-T27454-50mg50mg£1,661.00
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Quantity:
TAR-T27454-100mg100mg£2,079.00
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Quantity:
TAR-T27454-500mg500mg£4,006.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
GSK2008607 is a competitive inhibitor of rTbIPMK with respect to Ins(1,4,5)P3.
CAS:
1244644-50-5
Formula:
C31H28F3N7O3S2
Molecular Weight:
667.73
Pathway:
MAPK
Purity:
0.98
SMILES:
CC(C)c1nc(c(s1)-c1ccnc(Nc2ccc(nc2)N2CCOCC2)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Target:
Raf

References

Stellwagen JC, et al. Development of potent B-RafV600E inhibitors containing an arylsulfonamide headgroup. Bioorg Med Chem Lett. 2011;21(15):4436-4440. Adjabeng George, et al. Preparation of thiazole sulfonamide and oxazole sulfonamide kinase inhibitors for cancer treatment. WO2010104899 A1.