NS-2710
Code | Size | Price |
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TAR-T28197-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T28197-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T28197-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.
CAS:
184220-36-8
Formula:
C22H20N4O
Molecular Weight:
356.429
Purity:
0.98
SMILES:
CCON=C(/C)c1ccc2n(cnc2c1)-c1cccc(c1)-c1cccnc1
References
1. Atack JR. GABAA receptor subtype-selective modulators. I. ?2/?3-selective agonists as non-sedating anxiolytics. Curr Top Med Chem. 2011;11(9):1176-202. Review. PubMed PMID: 21050172.
2. Evenden J, Duncan B, Ko T. A comparison of the effects of psychotomimetics and anxiolytics on punished and unpunished responding maintained by fixed interval schedules of food reinforcement in the rat. Behav Pharmacol. 2006 Feb;17(1):87-99. PubMed PMID: 16377966.
3. Mirza NR, Nielsen E?. Do subtype-selective gamma-aminobutyric acid A receptor modulators have a reduced propensity to induce physical dependence in mice? J Pharmacol Exp Ther. 2006 Mar;316(3):1378-85. PubMed PMID: 16352707.
4. Atack JR. Anxioselective compounds acting at the GABA(A) receptor benzodiazepine binding site. Curr Drug Targets CNS Neurol Disord. 2003 Aug;2(4):213-32. Review. PubMed PMID: 12871032.