TargetMol

NVP ACQ090

Product Code:
 
TAR-T28220
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28220-5mg5mg£1,251.00
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TAR-T28220-50mg50mg£2,464.00
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Quantity:
TAR-T28220-100mg100mg£3,283.00
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This product comes from: United States.
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Further Information

Bioactivity:
NVP ACQ090 is a potent and subtype-selective somatostatin sst(3) receptor antagonist.
CAS:
362612-47-3
Formula:
C30H40F2N4O2
Molecular Weight:
526.673
Purity:
0.98
SMILES:
[H][C@@]12CCCC[C@]1([H])[C@@H](CN(CC(C)Cc1ccc(OC)nc1)C2)C(=O)N1CCN(CC1)c1ccc(F)c(F)c1

References

1. Lehmann A, Kliewer A, G?nther T, Nagel F, Schulz S. Identification of Phosphorylation Sites Regulating sst3 Somatostatin Receptor Trafficking. Mol Endocrinol. 2016 Jun;30(6):645-59. doi: 10.1210/me.2015-1244. Epub 2016 Apr 21. PubMed PMID: 27101376. 2. Einstein EB, Patterson CA, Hon BJ, Regan KA, Reddi J, Melnikoff DE, Mateer MJ, Schulz S, Johnson BN, Tallent MK. Somatostatin signaling in neuronal cilia is critical for object recognition memory. J Neurosci. 2010 Mar 24;30(12):4306-14. doi: 10.1523/JNEUROSCI.5295-09.2010. PubMed PMID: 20335466; PubMed Central PMCID: PMC3842454. 3. Troxler T, Hurth K, Schuh KH, Schoeffter P, Langenegger D, Enz A, Hoyer D. Decahydroisoquinoline derivatives as novel non-peptidic, potent and subtype-selective somatostatin sst(3) receptor antagonists. Bioorg Med Chem Lett. 2010 Mar 1;20(5):1728-34. doi: 10.1016/j.bmcl.2010.01.063. Epub 2010 Jan 21. PubMed PMID: 20137944.