Setastine

TargetMol
Product Code: TAR-T28761
Supplier: TargetMol
CodeSizePrice
TAR-T28761-5mg5mg£850.00
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Quantity:
TAR-T28761-50mg50mg£1,661.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T28761-100mg100mg£2,079.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Further Information

Bioactivity:
Setastine, a highly selective H1 receptor antagonist, acts as a non-sedative antihistamine.
CAS:
64294-95-7
Formula:
C22H28ClNO
Molecular Weight:
357.92
Purity:
0.98
SMILES:
CC(OCCN1CCCCCC1)(c1ccccc1)c1ccc(Cl)cc1

References

1. Xiu MG, Wang DF. [Observation on therapeutic effect of acupoint injection desensitization with autoblood on chronic urticaria]. Zhongguo Zhen Jiu. 2011 Jul;31(7):610-2. Chinese. PubMed PMID: 21823283. 2. Rajna P, Veres J. Assessing the sedative (adverse) effects of antiallergic drugs by quantitative electroencephalography: effects of setastine a non-sedating antihistaminic drug. Ther Hung. 1994;42(1):14-20. PubMed PMID: 7761959. 3. Herjavecz I, Kar?csonyi E, M?lbacher S, Radics K, Szil?gyi R, Gacs?lyi I. Comparative clinical examination of Loderix (setastinum) and astemizole in pollenosis. Ther Hung. 1993;41(4):141-5. PubMed PMID: 8029782. 4. Mer?tey K, Falus A, Taga T, Kishimoto T. Histamine influences the expression of the interleukin-6 receptor on human lymphoid, monocytoid and hepatoma cell lines. Agents Actions. 1991 May;33(1-2):189-91. PubMed PMID: 1680274.