Silperisone HCl
Code | Size | Price |
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TAR-T28778-1mg | 1mg | £177.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T28778-5mg | 5mg | £328.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T28778-10mg | 10mg | £456.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T28778-25mg | 25mg | £702.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T28778-50mg | 50mg | £938.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T28778-100mg | 100mg | £1,259.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T28778-500mg | 500mg | £2,448.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Silperisone is a sodium channel protein type 2 alpha channel blocker. Silperisone is a tolperisone like organosilicon compound with centrally acting muscle relaxant properties.
CAS:
140944-30-5
Formula:
C15H25ClFNSi
Molecular Weight:
301.91
Purity:
0.98
SMILES:
Cl.C[Si](C)(CN1CCCCC1)Cc1ccc(F)cc1
References
1. Lazar A, Lenkey N, Pesti K, Fodor L, Mike A. Different pH-sensitivity patterns of 30 sodium channel inhibitors suggest chemically different pools along the access pathway. Front Pharmacol. 2015 Sep 25;6:210. doi: 10.3389/fphar.2015.00210. PubMed PMID: 26441665; PubMed Central PMCID: PMC4585259.
2. Farkas S. Silperisone: a centrally acting muscle relaxant. CNS Drug Rev. 2006 Fall-Winter;12(3-4):218-35. Review. PubMed PMID: 17227288.
3. Kocsis P, Farkas S, Fodor L, Bielik N, Th?n M, Kolok S, Gere A, Csejtei M, Tarnawa I. Tolperisone-type drugs inhibit spinal reflexes via blockade of voltage-gated sodium and calcium channels. J Pharmacol Exp Ther. 2005 Dec;315(3):1237-46. PubMed PMID: 16126840.
4. Farkas S, Berzsenyi P, K?rp?ti E, Kocsis P, Tarnawa I. Simple pharmacological test battery to assess efficacy and side effect profile of centrally acting muscle relaxant drugs. J Pharmacol Toxicol Methods. 2005 Sep-Oct;52(2):264-73. PubMed PMID: 16125625.