ASP-4000 HCl
Code | Size | Price |
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TAR-T30166-5mg | 5mg | £1,010.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T30166-50mg | 50mg | £1,982.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T30166-100mg | 100mg | £2,560.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
ASP-4000 HCl is an inhibitor of dipeptidyl peptidase 4 (DPP) with anti-hyperglycemic activity.
CAS:
851389-35-0
Formula:
C12H18ClN3O2
Molecular Weight:
271.75
Purity:
0.98
SMILES:
Cl.O[C@@H]1C[C@@H]2C[C@H]1N[C@@H]2C(=O)N1CCC[C@H]1C#N
References
1. Tanaka-Amino K, Hatakeyama Y, Takakura S, Mutoh S. Constitutive increase in active GLP-1 levels by the DPP4 inhibitor ASP4000 on a new meal tolerance test in Zucker fatty rats. Pharmacol Res. 2009 Oct;60(4):264-9. doi: 10.1016/j.phrs.2009.03.018. Epub 2009 Apr 7. PubMed PMID: 19520592.
2. Tanaka-Amino K, Matsumoto K, Hatakeyama Y, Takakura S, Mutoh S. ASP4000, a slow-binding dipeptidyl peptidase 4 inhibitor, has antihyperglycemic activity of long duration in Zucker fatty rats. Acta Diabetol. 2010 Mar;47(1):43-8. doi: 10.1007/s00592-009-0096-5. Epub 2009 Feb 24. PubMed PMID: 19238312.
3. Tanaka-Amino K, Matsumoto K, Hatakeyama Y, Shima I, Takakura S, Muto S. ASP4,000, a novel, selective, dipeptidyl peptidase 4 inhibitor with antihyperglycemic activity. Eur J Pharmacol. 2008 Aug 20;590(1-3):444-9. doi: 10.1016/j.ejphar.2008.05.034. Epub 2008 Jun 24. PubMed PMID: 18582861.