BMS-694153

TargetMol
Product Code: TAR-T30537
Supplier: TargetMol
CodeSizePrice
TAR-T30537-5mg5mg£1,332.00
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Quantity:
TAR-T30537-50mg50mg£2,625.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T30537-100mg100mg£3,524.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Further Information

Bioactivity:
BMS-694153 is a potent and selective CGRP receptor antagonist.
CAS:
1050381-35-5
Formula:
C35H45FN8O3
Molecular Weight:
644.796
Purity:
0.98
SMILES:
Cc1cc(C[C@@H](NC(=O)N2CCC(CC2)N2Cc3cccc(F)c3NC2=O)C(=O)N2CCC(CC2)N2CCCCC2)cc2cn[nH]c12

References

1. Zheng N, Buzescu A, Pasas-Farmer S, Arnold ME, Ouyang Z, Jemal M, Peng Q, Van Vleet T, Zeng J. A simplified and completely automated workflow for regulated LC-MS/MS bioanalysis using cap-piercing direct sampling and evaporation-free solid phase extraction. J Chromatogr B Analyt Technol Biomed Life Sci. 2013 Mar 15;921-922:64-74. doi: 10.1016/j.jchromb.2013.01.028. Epub 2013 Feb 4. PubMed PMID: 23435343. 2. Luo G, Chen L, Pin SS, Xu C, Conway CM, Macor JE, Dubowchik GM. Calcitonin gene-related peptide (CGRP) receptor antagonists: novel aspartates and succinates. Bioorg Med Chem Lett. 2012 Apr 15;22(8):2912-6. doi: 10.1016/j.bmcl.2012.02.066. Epub 2012 Mar 3. PubMed PMID: 22429471. 3. Luo G, Chen L, Civiello R, Pin SS, Xu C, Kostich W, Kelley M, Conway CM, Macor JE, Dubowchik GM. Calcitonin gene-related peptide (CGRP) receptor antagonists: pyridine as a replacement for a core amide group. Bioorg Med Chem Lett. 2012 Apr 15;22(8):2917-21. doi: 10.1016/j.bmcl.2012.02.065. Epub 2012 Mar 3. PubMed PMID: 22429470. 4. Fischer MJ. Calcitonin gene-related peptide receptor antagonists for migraine. Expert Opin Investig Drugs. 2010 Jul;19(7):815-23. doi: 10.1517/13543784.2010.490829. Review. PubMed PMID: 20482328.