GLPG0634 analog

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TargetMol
Product Code: TAR-T3076
Supplier: TargetMol
CodeSizePrice
TAR-T3076-1mg1mg£98.00
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TAR-T3076-2mg2mg£109.00
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TAR-T3076-5mg5mg£135.00
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TAR-T3076-1mL1 mL * 10 mM (in DMSO)£142.00
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TAR-T3076-10mg10mg£189.00
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Quantity:
TAR-T3076-25mg25mg£293.00
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Quantity:
TAR-T3076-50mg50mg£464.00
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TAR-T3076-100mg100mg£627.00
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Quantity:
TAR-T3076-500mg500mg£1,235.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
GLPG0634 (analog) is a specific JAK1 inhibitor with IC50 of 10/28/810/116 nM for JAK1/2/3 and TYK2, respectively.
CAS:
1206101-20-3
Formula:
C23H18N6O2
Molecular Weight:
410.437
Pathway:
JAK/STAT signaling; Chromatin/Epigenetic; Stem Cells; Tyrosine Kinase/Adaptors; Angiogenesis
Purity:
0.9923
SMILES:
O=C(Nc1nc2cccc(-c3ccc(OCc4ccc(nc4)C#N)cc3)n2n1)C1CC1
Target:
Tyrosine Kinases; JAK

References

1. Van Rompaey L, et al. J Immunol. 2013, 191(7), 3568-3577.