CCG-257081

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TargetMol
Product Code: TAR-T30778
Supplier: TargetMol
CodeSizePrice
TAR-T30778-1mg1mg£174.00
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TAR-T30778-5mg5mg£322.00
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TAR-T30778-10mg10mg£445.00
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TAR-T30778-25mg25mg£686.00
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TAR-T30778-50mg50mg£930.00
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TAR-T30778-100mg100mg£1,235.00
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TAR-T30778-500mg500mg£2,384.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
CCG-257081 is an inihibitor of Rho/MRTF/SRF pathway. CCG-257081 has shown efficacy in preventing bleomycin-induced fibrosis in several mouse models.
CAS:
1922098-90-5
Formula:
C24H19ClF3N3O2
Molecular Weight:
473.88
Pathway:
GPCR/G Protein|Cell Cycle/Checkpoint|MAPK
Purity:
0.98
SMILES:
Fc1cc(cc(c1)-c1ccncc1)C(=O)N1CC(CC(F)(F)C1)C(=O)Nc1ccc(Cl)cc1
Target:
Rho|Ras

References

1. https://www.researchgate.net/grant/Demonstrating-the-feasibility-of-CCG-257081-as-a-preventive-therapy-to-inhibit-bleomycin-induced-lung-fibrosis-in-mice_3433689