Cgp 55802A
| Code | Size | Price |
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| TAR-T30840-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
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Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Documents
Further Information
Bioactivity:
CGP 55802A is a novel photoaffinity ligand for in-situ labeling of NMDA receptors.
CAS:
152564-63-1
Formula:
C18H24IN5NaO7P
Molecular Weight:
603.286
Purity:
0.98
SMILES:
[Na+].NC(C=C(/CCCCCCNC(=O)c1ccc(N=[N+]=[N-])c(I)c1O)CP(O)(O)=O)C([O-])=O
References
1. Resink A, Villa M, Benke D, M?hler H, Bal?zs R. Regulation of the expression of NMDA receptor subunits in rat cerebellar granule cells: effect of chronic K(+)-induced depolarization and NMDA exposure. J Neurochem. 1995 Feb;64(2):558-65. PubMed PMID: 7830048.
2. Heckendorn R, Allgeier H, Baud J, Gunzenhauser W, Angst C. Synthesis and binding properties of 2-amino-5-phosphono-3-pentenoic acid photoaffinity ligands as probes for the glutamate recognition site of the NMDA receptor. J Med Chem. 1993 Nov 12;36(23):3721-6. PubMed PMID: 7902441.
3. Marti T, Benke D, Mertens S, Heckendorn R, Pozza M, Allgeier H, Angst C, Laurie D, Seeburg P, Mohler H. Molecular distinction of three N-methyl-D-aspartate-receptor subtypes in situ and developmental receptor maturation demonstrated with the photoaffinity ligand 125I-labeled CGP 55802A. Proc Natl Acad Sci U S A. 1993 Sep 15;90(18):8434-8. PubMed PMID: 8378316; PubMed Central PMCID: PMC47371.
4. Benke D, Marti T, Heckendorn R, Rehm H, K?nzi R, Allgeier H, Angst C, Mohler H. Photoaffinity labeling of the NMDA receptor. Eur J Pharmacol. 1993 Jul 15;246(2):179-80. PubMed PMID: 8375463.