CI 992
Code | Size | Price |
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TAR-T30921-5mg | 5mg | £1,733.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T30921-50mg | 50mg | £3,428.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T30921-100mg | 100mg | £4,729.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
CI 992 is a novel potent inhibitor of primate renin.
CAS:
135704-06-2
Formula:
C33H52N6O7S2
Molecular Weight:
708.93
Purity:
0.98
SMILES:
CC(C)C[C@H](O)[C@H](O)[C@H](CC1CCCCC1)N[C@@H](Cc1csc(N)n1)C(=O)NC(=O)[C@H](Cc1ccccc1)NS(=O)(=O)N1CCOCC1
References
1. Cook JA, Burger PJ, Michniewicz BM, Nordblom GD, Hicks GW, Kaplan C, Ryan MJ. Pharmacokinetics and pharmacodynamics of CI-992 following intravenous and oral administration to cynomolgus monkeys. Biopharm Drug Dispos. 1998 Apr;19(3):185-91. PubMed PMID: 9570002.
2. Ryan MJ, Hicks GW, Batley BL, Rapundalo ST, Patt WC, Taylor DG, Keiser JA. Effect of an orally active renin inhibitor Cl-992 on blood pressure in normotensive and hypertensive monkeys. J Pharmacol Exp Ther. 1994 Jan;268(1):372-9. PubMed PMID: 8301578.