CPFPX
| Code | Size | Price |
|---|
| TAR-T31086-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Documents
Further Information
Bioactivity:
CPFPX is a highly selective radioactive ligand for the A1 adenosine receptor (A1AR).
CAS:
227205-79-0
Formula:
C16H23FN4O2
Molecular Weight:
321.387
Purity:
0.98
SMILES:
CCCn1c(=O)n(CCC[18F])c2nc([nH]c2c1=O)C1CCCC1
References
1. Kroll T, Elmenhorst D, Weisshaupt A, Beer S, Bauer A. Reproducibility of non-invasive a1 adenosine receptor quantification in the rat brain using [(18)F]CPFPX and positron emission tomography. Mol Imaging Biol. 2014 Oct;16(5):699-709. doi: 10.1007/s11307-014-0729-0. PubMed PMID: 24595700.
2. Elmenhorst D, Kroll T, Wedekind F, Weisshaupt A, Beer S, Bauer A. In vivo kinetic and steady-state quantification of 18F-CPFPX binding to rat cerebral A1 adenosine receptors: validation by displacement and autoradiographic experiments. J Nucl Med. 2013 Aug;54(8):1411-9. doi: 10.2967/jnumed.112.115576. PubMed PMID: 23740103.
3. Elmenhorst D, Meyer PT, Matusch A, Winz OH, Bauer A. Caffeine occupancy of human cerebral A1 adenosine receptors: in vivo quantification with 18F-CPFPX and PET. J Nucl Med. 2012 Nov;53(11):1723-9. doi: 10.2967/jnumed.112.105114. PubMed PMID: 22966134.