Denagliptin tosylate
Code | Size | Price |
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TAR-T31378-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T31378-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T31378-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Denagliptin (GW823093 or GSK-823093) is a dipeptidyl peptidase IV (DPP-IV) inhibitor.
CAS:
811432-66-3
Formula:
C27H26F3N3O4S
Molecular Weight:
545.58
Purity:
0.98
SMILES:
Cc1ccc(cc1)S(O)(=O)=O.N[C@@H](C(c1ccc(F)cc1)c1ccc(F)cc1)C(=O)N1C[C@@H](F)C[C@H]1C#N
References
1. De Serres M, Bowers G, Boyle G, Beaumont C, Castellino S, Sigafoos J, Dave M, Roberts A, Shah V, Olson K, Patel D, Wagner D, Yeager R, Serabjit-Singh C. Evaluation of a chimeric (uPA+/+)/SCID mouse model with a humanized liver for prediction of human metabolism. Xenobiotica. 2011 Jun;41(6):464-75. doi: 10.3109/00498254.2011.560295. Epub 2011 Mar 4. PubMed PMID: 21370990.
2. Joshi BK, Ramsey B, Johnson B, Patterson DE, Powers J, Facchine KL, Osterhout M, Leblanc MP, Bryant-Mills R, Copley RC, Sides SL. Elucidating the pathways of degradation of denagliptin. J Pharm Sci. 2010 Jul;99(7):3030-40. doi: 10.1002/jps.22069. PubMed PMID: 20112433.