TargetMol

Enadoline hydrochloride

Product Code:
 
TAR-T31621
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T31621-5mg5mg£1,010.00
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TAR-T31621-50mg50mg£1,982.00
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Quantity:
TAR-T31621-100mg100mg£2,560.00
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This product comes from: United States.
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Further Information

Bioactivity:
Enadoline Hydrochloride is a highly selective κ-opioid agonist that may be developed as an analgesic.
CAS:
124439-07-2
Formula:
C24H33ClN2O3
Molecular Weight:
432.99
Purity:
0.98
SMILES:
Cl.CN([C@H]1CC[C@@]2(CCCO2)C[C@@H]1N1CCCC1)C(=O)Cc1cccc2occc12

References

1. Walsh SL, Strain EC, Abreu ME, Bigelow GE. Enadoline, a selective kappa opioid agonist: comparison with butorphanol and hydromorphone in humans. Psychopharmacology (Berl). 2001 Sep;157(2):151-62. PubMed PMID: 11594439. 2. Walsh SL, Geter-Douglas B, Strain EC, Bigelow GE. Enadoline and butorphanol: evaluation of kappa-agonists on cocaine pharmacodynamics and cocaine self-administration in humans. J Pharmacol Exp Ther. 2001 Oct;299(1):147-58. PubMed PMID: 11561074. 3. Carey GJ, Bergman J. Enadoline discrimination in squirrel monkeys: effects of opioid agonists and antagonists. J Pharmacol Exp Ther. 2001 Apr;297(1):215-23. PubMed PMID: 11259547. 4. Hinton JP, Hudson G. Unbound plasma concentrations may predict neuroprotective brain concentrations: a brain microdialysis and pharmacokinetic study of enadoline in rats. Acta Neurochir Suppl. 1999;75:7-9. PubMed PMID: 10635368.