GYKI-46903 HCl
Code | Size | Price |
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TAR-T32033-5mg | 5mg | £1,010.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T32033-50mg | 50mg | £1,982.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T32033-100mg | 100mg | £2,560.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
GYKI-46903 is a noncompetitive 5-HT3 receptor antagonist.
CAS:
142999-59-5
Formula:
C17H21ClFNO2
Molecular Weight:
325.81
Purity:
0.98
SMILES:
Cl.CCC(=O)O[C@@H]1CCN2CC=C([C@@H]1C2)c1ccc(F)cc1
References
1. Maksay G, B?r? T, Bugovics G. Allosteric modulation of 5-HT3 serotonin receptors. Eur J Pharmacol. 2005 May 2;514(1):17-24. Epub 2005 Apr 22. PubMed PMID: 15878320.
2. Vit?lis B, Sebesty?n L, Sike M, S?lyom S, H?rsing LG Jr. Binding characteristics of GYKI-46 903, a non-competitive ligand at 5-HT3 receptors. Pharmacol Res. 2001 Mar;43(3):291-9. PubMed PMID: 11401422.
3. Bagdy E, Solyom S, Harsing LG Jr. Feedback stimulation of somatodendritic serotonin release: a 5-HT3 receptor-mediated effect in the raphe nuclei of the rat. Brain Res Bull. 1998;45(2):203-8. PubMed PMID: 9443841.
4. Csillik-Perczel V, Bakonyi A, Yemane T, Vitalis B, Horvath E, Solyom S, Szekely JI, Harsing LG Jr. GYKI-46 903, a non-competitive antagonist for 5-HT3 receptors. Pharmacol Toxicol. 1996 Jul;79(1):32-9. PubMed PMID: 8841094.