Mdl 28564
| Code | Size | Price |
|---|
| TAR-T33264-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Documents
Further Information
Bioactivity:
Mdl 28564 is a neurokinin A analog.
CAS:
127370-75-6
Formula:
C35H58N8O9
Molecular Weight:
734.896
Purity:
0.98
SMILES:
CC(C)C[C@@H](CN[C@@H](CC(C)C)C(N)=O)N(CC(N)=O)C(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(O)=O)C(C)C
References
Maggi CA, Patacchini R, Eglezos A, Quartara L, Giuliani S, Giachetti A. Tachykinin receptors in the guinea-pig renal pelvis: activation by exogenous and endogenous tachykinins. Br J Pharmacol. 1992 Sep;107(1):27-33. PubMed PMID: 1384907; PubMed Central PMCID: PMC1907585.
Buck SH, Harbeson SL, Hassmann CF 3rd, Shatzer SA, Rouissi N, Nantel F, van Giersbergen PL. [Leu9 psi(CH2NH)Leu10]-neurokinin A (4-10) (MDL 28,564) distinguishes tissue tachykinin peptide NK2 receptors. Life Sci. 1990;47(10):PL37-41. PubMed PMID: 2170788.
Giuliani S, Patacchini R, Barbanti G, Turini D, Rovero P, Quartara L, Giachetti A, Maggi CA. Characterization of the tachykinin neurokinin-2 receptor in the human urinary bladder by means of selective receptor antagonists and peptidase inhibitors. J Pharmacol Exp Ther. 1993 Nov;267(2):590-5. PubMed PMID: 8246132.
Patacchini R, Astolfi M, Quartara L, Rovero P, Giachetti A, Maggi CA. Further evidence for the existence of NK2 tachykinin receptor subtypes. Br J Pharmacol. 1991 Sep;104(1):91-6. PubMed PMID: 1664768; PubMed Central PMCID: PMC1908267.