MK-0952 Sodium

TargetMol
Product Code: TAR-T33424L
Supplier: TargetMol
CodeSizePrice
TAR-T33424L-5mg5mg£930.00
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Quantity:
TAR-T33424L-50mg50mg£1,821.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T33424L-100mg100mg£2,319.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Further Information

Bioactivity:
MK-0952 Sodium is a salt form of MK-0952, which is a selective PDE4 inhibitor.
CAS:
934995-88-7
Formula:
C28H21FN3NaO4
Molecular Weight:
505.481
Purity:
0.98
SMILES:
[Na+].[O-]C(=O)C1CC1c1ccc(cc1F)-c1cccc(c1)-n1cc(C(=O)NC2CC2)c(=O)c2cccnc12

References

Heckman PR, Wouters C, Prickaerts J. Phosphodiesterase inhibitors as a target for cognition enhancement in aging and Alzheimer's disease: a translational overview. Curr Pharm Des. 2015;21(3):317-31. Review. PubMed PMID: 25159073. Gallant M, Aspiotis R, Day S, Dias R, Dub? D, Dub? L, Friesen RW, Girard M, Guay D, Hamel P, Huang Z, Lacombe P, Lalibert? S, L?vesque JF, Liu S, Macdonald D, Mancini J, Nicholson DW, Styhler A, Townson K, Waters K, Young RN, Girard Y. Discovery of MK-0952, a selective PDE4 inhibitor for the treatment of long-term memory loss and mild cognitive impairment. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6387-93. doi: 10.1016/j.bmcl.2010.09.087. Epub 2010 Sep 21. PubMed PMID: 20933411.