Inupadenant

TargetMol
Product Code: TAR-T37014
Supplier: TargetMol
CodeSizePrice
TAR-T37014-5mg5mg£1,026.00
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Quantity:
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Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Further Information

Bioactivity:
Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].
CAS:
2246607-08-7
Formula:
C25H26F2N8O4S2
Molecular Weight:
604.65
Purity:
0.98
SMILES:
N/A

References

Laurence Buisseret, et al. Phase 1 trial of the adenosine A2Areceptor antagonist inupadenant (EOS-850): Update on tolerability, and antitumor activity potentially associated with the expression of the A2A receptor within the tumor. Journal of Clinical Oncology. Volume 39, Issue 15_suppl.