PF-03622905
Code | Size | Price |
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TAR-T38461-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
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Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
PF-03622905 is a potent and ATP-competitive PKC inhibitor with IC 50 s of 5.6 nM, 14.5 nM, 13 nM, 37.7 nM, and 74.1 nM for PKCα , PKCβI , PKCβII , PKCγ , and PKC? , respectively. PF-03622905 shows high specificity for PKC over other protein kinases.
CAS:
1072100-15-2
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0
References
Stephan Grant, et al. Discovery of a novel class of targeted kinase inhibitors that blocks protein kinase C signaling and ameliorates retinal vascular leakage in a diabetic rat model. Eur J Pharmacol. 2010 Feb 10;627(1-3):16-25.