ALK-IN-12
| Code | Size | Price |
|---|
| TAR-T38584-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Documents
Further Information
Bioactivity:
ALK-IN-12 is a potent and orally active ALK inhibitor with an IC 50 of 0.18 nM. ALK-IN-12 also inhibits IGF1R and InsR (IC 50 =20.3 and 90.6 nM). Antitumor activities.
CAS:
1197958-53-4
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0
References
Huang WS, et al. Discovery of Brigatinib (AP26113), a Phosphine Oxide-Containing, Potent, Orally Active Inhibitor of Anaplastic Lymphoma Kinase. J Med Chem. 2016;59(10):4948-4964.