EZH2-IN-4
| Code | Size | Price |
|---|
| TAR-T39497-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Documents
Further Information
Bioactivity:
EZH2-IN-4 is an orally active, potent EZH2 inhibitor with IC 50 s of 0.923 nM and 2.65 nM against wild type (WT) 5-membered (5-mer) EZH2 and mutant 5-mer EZH2, respectively. EZH2-IN-4 has anti-cancer activity.
CAS:
2088132-99-2
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0
References
Esteban DOMINGUEZ, et al. Inhibitors of ezh2. WO2017035060A1.