CDK12-IN-4
| Code | Size | Price |
|---|
| TAR-T40288-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Documents
Further Information
Bioactivity:
CDK12-IN-4, a pyrazolotriazine, is a potent CDK12 inhibitor with an IC 50 of 0.641 μM at high ATP (2 mM). CDK12-IN-4 has no effect on CDK2/Cyclin E (IC 50 >20 μM) and CDK9/Cyclin T1 (IC 50 >20 μM) at high ATP (2 mM) (WO2021116178A1).
CAS:
2651196-69-7
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0
References
Kai Thede, et al. Pyrazolotriazines. WO2021116178A1.