TargetMol

CDK12-IN-6

Product Code:
 
TAR-T40289
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

No additional charges, what you see is what you pay! *

CodeSizePrice
TAR-T40289-5mg5mg£850.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
Prices exclude any Taxes / VAT
How to order with us   Contact us
Stay in control of your spending. These prices have no additional charges, not even shipping!
* Rare exceptions are clearly labelled (only 0.14% of items!).
Multibuy discounts available! Contact us to find what you can save.
This product comes from: United States.
Typical lead time: 10-14 working days.
Contact us for more accurate information.
  • Further Information
  • Documents
  • References
  • Show All

Further Information

Bioactivity:
CDK12-IN-6, a pyrazolotriazine, is a potent CDK12 inhibitor with an IC 50 of 1.19 μM at high ATP (2 mM). CDK12-IN-6 has no effect on CDK2/Cyclin E (IC 50 >20 μM) and CDK9/Cyclin T1 (IC 50 >20 μM) at high ATP (2 mM) (WO2021116178A1).
CAS:
2651196-71-1
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0

References

Kai Thede, et al. Pyrazolotriazines. WO2021116178A1.