CDK12-IN-5
| Code | Size | Price |
|---|
| TAR-T40290-5mg | 5mg | £410.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
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Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Documents
Further Information
Bioactivity:
CDK12-IN-5, a pyrazolotriazine, is a potent CDK12 inhibitor with an IC 50 of 23.9 nM at high ATP (2 mM). CDK12-IN-5 has no effect on CDK2/Cyclin E (IC 50 =173 μM) and CDK9/Cyclin T1 (IC 50 =127 μM) at high ATP (2 mM) (WO2021116178A1).
CAS:
2651200-35-8
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0
References
Kai Thede, et al. Pyrazolotriazines. WO2021116178A1.