AR-M 1000390 hydrochloride
Code | Size | Price |
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TAR-T4236-5mg | 5mg | £122.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
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Quantity:
TAR-T4236-1mL | 1 mL * 10 mM (in DMSO) | £127.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T4236-10mg | 10mg | £156.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T4236-25mg | 25mg | £246.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T4236-50mg | 50mg | £389.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T4236-100mg | 100mg | £548.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
AR-M 1000390 (hydrochloride), also known as ARM-390, is a low-internalizing nonpeptidic δ-selective opioid receptor agonist; derivative of SNC 80. Does not trigger acute desensitization of the analgesic response; reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration.
CAS:
209808-47-9
Formula:
C23H29ClN2O
Molecular Weight:
384.95
Pathway:
GPCR/G Protein; Neuroscience; Endocrinology/Hormones
Purity:
0.9968
SMILES:
Cl.CCN(CC)C(=O)c1ccc(cc1)C(=C1CCNCC1)c1ccccc1
Target:
Opioid Receptor
References
Marie N,etal.Pharmacological characterization of AR-M1000390 at human delta opioid receptors.Life Sci. 2003 Aug 15;73(13):1691-704.
Pradhan AA,etal.Ligand-directed trafficking of the ?-opioid receptor in vivo: two paths toward analgesic tolerance.J Neurosci. 2010 Dec 8;30(49):16459-68.