ARN272

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TargetMol
Product Code: TAR-T5357
Supplier: TargetMol
CodeSizePrice
TAR-T5357-5mg5mg£102.00
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TAR-T5357-1mL1 mL * 10 mM (in DMSO)£105.00
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TAR-T5357-10mg10mg£122.00
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TAR-T5357-25mg25mg£168.00
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TAR-T5357-50mg50mg£230.00
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TAR-T5357-100mg100mg£367.00
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TAR-T5357-200mg200mg£511.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).
CAS:
488793-85-7
Formula:
C27H20N4O2
Molecular Weight:
432.483
Pathway:
Metabolism; Neuroscience
Purity:
0.9823
SMILES:
Oc1ccc(cc1)-c1n[nH]c(=N/c2ccc(cc2)C(=O)Nc2ccccc2)c2ccccc12
Target:
FAAH

References

O'Brien LD, et al. Anandamide transport inhibition by ARN272 attenuates nausea-induced behaviour in rats, and vomiting in shrews (Suncus murinus). Br J Pharmacol. 2013 Nov;170(5):1130-6. Fu J, et al. A catalytically silent FAAH-1 variant drives anandamide transport in neurons. Nat Neurosci. 2011 Nov 20;15(1):64-9.