TAK-700

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TargetMol
Product Code: TAR-T6050
Supplier: TargetMol
CodeSizePrice
TAR-T6050-1mg1mg£98.00
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TAR-T6050-2mg2mg£109.00
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TAR-T6050-5mg5mg£135.00
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TAR-T6050-1mL1 mL * 10 mM (in DMSO)£142.00
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TAR-T6050-10mg10mg£182.00
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TAR-T6050-25mg25mg£294.00
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TAR-T6050-50mg50mg£430.00
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TAR-T6050-100mg100mg£589.00
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TAR-T6050-200mg200mg£784.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
TAK-700 (Orteronel) is a potent and highly selective human 17, 20-lyase inhibitor with IC50 of 38 nM, exhibits >1000-fold selectivity over other CYPs (e.g. 11-hydroxylase and CYP3A4). Phase 3.
CAS:
426219-18-3
Formula:
C18H17N3O2
Molecular Weight:
307.353
Pathway:
Metabolism
Purity:
0.9975
SMILES:
CNC(=O)c1ccc2cc(ccc2c1)C1(O)CCn2cncc12
Target:
P45

References

Kaku T, et al. Bioorg Med Chem. 2011, 19(21), 6383-6399. Yamaoka M, et al. J Steroid Biochem Mol Biol. 2012, 129(3-5), 115-128.