Desmethyl Erlotinib

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TargetMol
Product Code: TAR-T6328
Supplier: TargetMol
CodeSizePrice
TAR-T6328-1mg1mg£109.00
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TAR-T6328-2mg2mg£127.00
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TAR-T6328-5mg5mg£164.00
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TAR-T6328-1mL1 mL * 10 mM (in DMSO)£174.00
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TAR-T6328-10mg10mg£230.00
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TAR-T6328-25mg25mg£351.00
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TAR-T6328-50mg50mg£491.00
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TAR-T6328-100mg100mg£679.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
OSI-420 is the active metabolite of Erlotinib (EGFR inhibitor with IC50 of 2 nM).
CAS:
183321-86-0
Formula:
C21H21N3O4
Molecular Weight:
379.416
Pathway:
Metabolism; JAK/STAT signaling; Tyrosine Kinase/Adaptors; Angiogenesis
Purity:
0.9862
SMILES:
COCCOc1cc2ncnc(Nc3cccc(c3)C#C)c2cc1OCCO
Target:
EGFR; Drug Metabolite

References

Meany HJ, et al. Cancer Chemother Pharmacol. 2008, 62(3), 387-392. Moyer JD, et al. Cancer Res. 1997, 57(21), 4838-4848.